SCHEMBL9526274

SCHEMBL9526274

CC(C)(C)OC(=O)NCCC(=O)NCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
CYP3A4 P08684 4/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HTT P42858 3/20 0.38
CYP1A2 P05177 3/20 0.37
CYP2C19 P33261 3/20 0.37
KDM4E B2RXH2 1/20 0.37
ALOX15 P16050 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524354 0.94 NPC1 (0.44) NPC1RAB9ACKS1BSKP1SKP2
SCHEMBL9527984 0.83 SMN1; SMN2 (0.46) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL9525795 0.83 SMN1; SMN2 (0.46) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL9525116 0.80 SMN1; SMN2 (0.46) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL9407533 0.78 NPC1 (0.46) NPC1RAB9ASMN1; SMN2CYP3A4POLB
SCHEMBL9525433 0.78 EPHX1 (0.45) NPC1SMN1; SMN2POLBALDH1A1CYP1A2
SCHEMBL9407563 0.78 NPC1 (0.41) NPC1RAB9ASMN1; SMN2CYP3A4POLB
SCHEMBL9524002 0.78 NPC1 (0.44) NPC1RAB9ASMN1; SMN2CYP3A4POLB
SCHEMBL9524919 0.77 HTT (0.51) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL9525530 0.76 HTT (0.46) NPC1RAB9ASMN1; SMN2CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed