SCHEMBL9525795

SCHEMBL9525795

NCCC(=O)NCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
POLB P06746 2/20 0.45
ADRA2C P18825 1/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HTT P42858 3/20 0.43
ALOX15 P16050 1/20 0.43
KDM4E B2RXH2 1/20 0.41
EGFR P00533 1/20 0.40
HCAR2 Q8TDS4 1/20 0.39
MAPK1 P28482 2/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 1/20 0.38
GAA P10253 1/20 0.38
GLA P06280 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527984 0.91 SMN1; SMN2 (0.46) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9525116 0.87 SMN1; SMN2 (0.46) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9524204 0.86 ADRA2C (0.52) SMN1; SMN2POLBADRA2CNPC1RAB9A
SCHEMBL9524919 0.84 HTT (0.51) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9526274 0.83 NPC1 (0.40) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9525706 0.83 CYP1A2 (0.41) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9525433 0.81 EPHX1 (0.45) SMN1; SMN2POLBNPC1ALDH1A1KDM4E
SCHEMBL9524354 0.80 NPC1 (0.44) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9524791 0.80 NPC1 (0.49) SMN1; SMN2POLBNPC1RAB9AALDH1A1
SCHEMBL9407533 0.79 NPC1 (0.46) SMN1; SMN2POLBNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed