SCHEMBL9525433

SCHEMBL9525433

O=C(CCNC(=O)Nc1cccc2ccccc12)NCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.45
TRPV1 Q8NER1 4/20 0.41
KDM4E B2RXH2 4/20 0.41
GSK3B P49841 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
NPY5R Q15761 1/20 0.39
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.38
KDR P35968 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525706 0.93 CYP1A2 (0.41) EPHX1SMN1; SMN2ALDH1A1CYP1A2CYP2C19
SCHEMBL9528510 0.92 SMN1; SMN2 (0.40) EPHX1SMN1; SMN2ALDH1A1CYP1A2CYP2C19
SCHEMBL9525362 0.86 BLM (0.43) SMN1; SMN2ALDH1A1CYP1A2CYP2C19KDR
SCHEMBL9524016 0.86 ALDH1A1 (0.41) EPHX1TRPV1KDM4EGSK3BSMN1; SMN2
SCHEMBL9524974 0.85 ALDH1A1 (0.41) TRPV1SMN1; SMN2ALDH1A1HSD17B10KDR
SCHEMBL9525424 0.84 ALDH1A1 (0.43) EPHX1TRPV1SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL9525236 0.84 ALDH1A1 (0.40) TRPV1KDM4ESMN1; SMN2ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL9526588 0.82 EPHX1 (0.46) EPHX1TRPV1KDM4EGSK3BL3MBTL1
SCHEMBL9527984 0.81 SMN1; SMN2 (0.46) KDM4ESMN1; SMN2ALDH1A1NPC1MAPT
SCHEMBL9525795 0.81 SMN1; SMN2 (0.46) KDM4ESMN1; SMN2ALDH1A1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed