SCHEMBL9526399

SCHEMBL9526399

OC(c1ccncc1)c1ccccc1C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CYP3A4 P08684 2/20 0.39
CYP17A1 P05093 2/20 0.39
CYP19A1 P11511 2/20 0.39
CYP11B2 P19099 2/20 0.39
CYP11B1 P15538 1/20 0.39
GAA P10253 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
IDO1 P14902 5/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9487949 0.86 MEN1 (0.43) ADRA2AADRA2BADRA2CGAACYP1A2
SCHEMBL23003623 0.73 CYP3A4 (0.48) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL11360995 0.72 ADRA2A (0.37) ADRA2AADRA2BADRA2CCYP3A4SLC6A2
SCHEMBL23882867 0.72 CYP3A4 (0.43) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL23882860 0.72 CYP3A4 (0.43) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL30251473 0.72 CYP3A4 (0.43) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL23882759 0.72 HDAC4 (0.47) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL23882758 0.72 HDAC4 (0.47) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL9528623 0.72 GAA (0.67) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1
SCHEMBL9526348 0.72 CYP11B1 (0.52) CYP3A4CYP17A1CYP19A1CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231996-B1 NOVEL AMINO ACID DERIVATIVES NOVO NORDISK A/S (DK) 1993-10-06 EP disclosed
EP-0231996-A2 Novel amino acid derivatives NOVO NORDISK A/S (DK) 1987-08-12 EP disclosed