SCHEMBL9526678

SCHEMBL9526678

O=C(NC1=NN(c2c(Cl)cc(C(F)(F)F)cc2Cl)C(=O)C1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.55
KMT2A Q03164 5/20 0.55
MAPT P10636 4/20 0.55
POLB P06746 3/20 0.55
RECQL P46063 3/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
THRB P10828 1/20 0.55
HTT P42858 1/20 0.55
P2RX1 P51575 1/20 0.50
GAA P10253 6/20 0.49
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KCNK3 O14649 1/20 0.44
LMNA P02545 2/20 0.43
MRGPRX4 Q96LA9 1/20 0.42
TRPA1 O75762 1/20 0.42
CYP1A2 P05177 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KCNH2 Q12809 1/20 0.42
GRK5 P34947 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10875014 0.88 MEN1 (0.68) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL124737 0.76 MEN1 (0.72) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL10867193 0.74 KMT2A (0.74) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL10061485 0.74 MAPT (0.55) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL11049234 0.72 MEN1 (0.70) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL9727104 0.72 P2RX1 (0.50) MEN1KMT2AMAPTPOLBP2RX1
SCHEMBL11047439 0.72 MEN1 (0.72) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL3190354 0.71 MAPT (0.53) MEN1KMT2AMAPTPOLBRECQL
SCHEMBL9525446 0.71 TDP1 (0.43) MEN1KMT2AMAPTL3MBTL1GAA
SCHEMBL10873637 0.70 KMT2A (0.56) MEN1KMT2AMAPTPOLBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274642-B1 HERBICIDAL AND FUNGICIDAL AGENTS BASED ON SUBSTITUTED PYRAZOLIN-5-ONE DERIVATIVES BAYER AG (DE) 1993-08-11 EP disclosed
US-5162528-A Pre- and post-emergence; phytaphthora in tomato plants; rice and wheat BAYER AKTIENGESELLSCHAFT (DE) 1992-11-10 US disclosed
US-5028717-A Herbicidal and fungicidal agents based on substituted pyrazolin-5-one derivatives BAYER AKTIENGESELLSCHAFT (DE) 1991-07-02 US disclosed
US-4909827-A Containing a C6-10 aryl group substituted in position 1 BAYER AKTIENGESELLSCHAFT (DE) 1990-03-20 US disclosed