SCHEMBL9526983

SCHEMBL9526983

O=C(CCCCl)Nc1ccnn1-c1c(Cl)cc(C(F)(F)F)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
GABRA2 P47869 7/20 0.39
GABRB2 P47870 7/20 0.39
LMNA P02545 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RHOC P08134 1/20 0.38
RHOA P61586 1/20 0.38
ALDH1A1 P00352 2/20 0.37
GABRB3 P28472 8/20 0.37
GABRP O00591 3/20 0.37
GABRD O14764 3/20 0.37
GABRA1 P14867 3/20 0.37
GABRB1 P18505 3/20 0.37
GABRG2 P18507 3/20 0.37
GABRA5 P31644 3/20 0.37
GABRA3 P34903 3/20 0.37
GABRA4 P48169 3/20 0.37
GABRE P78334 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10372959 0.89 BACE1 (0.43) BACE1GABRA2GABRB2LMNAALDH1A1
SCHEMBL9822782 0.85 GABRB3 (0.45) BACE1GABRA2GABRB2ALDH1A1GABRB3
SCHEMBL10560567 0.82 SMN1; SMN2 (0.43) BACE1GABRA2GABRB2LMNAALDH1A1
SCHEMBL10668017 0.79 MAPT (0.50) LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL10411191 0.79 BACE1 (0.39) BACE1GABRA2GABRB2RHOCRHOA
SCHEMBL10563948 0.78 BACE1 (0.40) BACE1GABRA2GABRB2LMNANPSR1
SCHEMBL9527645 0.78 BACE1 (0.42) BACE1GABRA2GABRB2GABRB3GABRP
SCHEMBL10388695 0.75 MAPT (0.37) HDAC1HDAC8GABRA2GABRB2NPSR1
SCHEMBL10400135 0.75 BACE1 (0.42) BACE1GABRA2GABRB2NPSR1ALDH1A1
SCHEMBL10668725 0.75 TSHR (0.50) BACE1NPSR1ALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0392241-B1 SUBSTITUTED 1-ARYLPYRAZOLS BAYER AG (DE) 1993-06-02 EP disclosed
US-4971989-A PESTICIDES, MITICIDES, INSECTICIDES AND NEMATOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1990-11-20 US disclosed
EP-0392241-A1 Substituted 1-Arylpyrazols BAYER AG (DE) 1990-10-17 EP disclosed