SCHEMBL9527149

SCHEMBL9527149

O=C(OCl)C1OC1c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.49
ALDH1A1 P00352 4/20 0.41
TSHR P16473 2/20 0.41
CES1 P23141 2/20 0.40
CES2 O00748 1/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 2/20 0.38
GAA P10253 1/20 0.38
F13A1 P00488 1/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CRHBP P24387 1/20 0.37
ATM Q13315 1/20 0.37
CRHR2 Q13324 1/20 0.37
TLR9 Q9NR96 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691641 0.85 EPHX1 (0.52) EPHX1ALDH1A1TSHRPOLBMAPK1
SCHEMBL8746385 0.81 TSHR (0.67) EPHX1ALDH1A1TSHRPOLBGAA
SCHEMBL8746369 0.80 EPHX1 (0.53) EPHX1ALDH1A1TSHRCES1CES2
SCHEMBL8746368 0.80 EPHX1 (0.53) EPHX1ALDH1A1TSHRCES1CES2
SCHEMBL8746372 0.80 EPHX1 (0.53) EPHX1ALDH1A1TSHRCES1CES2
SCHEMBL9525910 0.79 TSHR (0.46) EPHX1ALDH1A1TSHRPOLBGAA
SCHEMBL7112280 0.76 EPHX1 (0.68) EPHX1ALDH1A1CES1CES2TDP1
SCHEMBL11693135 0.74 EPHX1 (0.61) EPHX1ALDH1A1TSHRCES1CES2
SCHEMBL7405432 0.72 KMT2A (0.58) ALDH1A1GAAKMT2A
SCHEMBL29897104 0.71 EPHX1 (0.47) EPHX1ALDH1A1POLBMAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153229-B1 1-DETHIA 2-THIA-CEPHALOSPORANIC ACID DERIVATIVES, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS THERAPEUTIC AGENTS AND THE COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-07 EP disclosed
EP-0153229-A2 1-Dethia 2-thia-cephalosporanic acid derivatives, process and intermediates for their preparation, their use as therapeutic agents and the compositions containing them ROUSSEL-UCLAF (FR) 1985-08-28 EP disclosed