SCHEMBL9527201

SCHEMBL9527201

CC(=O)Nc1ccc2[nH]c3c(c2c1)Cc1ccccc1-3

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
MTNR1A P48039 2/20 0.60
MTNR1B P49286 2/20 0.60
KMT2A Q03164 1/20 0.60
MAOA P21397 2/20 0.56
CYP1A2 P05177 1/20 0.56
ADRA2A P08913 1/20 0.56
SLC6A2 P23975 1/20 0.56
HTR2C P28335 1/20 0.56
SLC6A4 P31645 1/20 0.56
HTR2B P41595 1/20 0.56
CA1 P00915 3/20 0.56
CA2 P00918 3/20 0.56
CA4 P22748 3/20 0.56
CA6 P23280 3/20 0.56
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
PARP1 P09874 4/20 0.49
ALDH1A1 P00352 1/20 0.48
ESR1 P03372 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527759 0.86 CA1 (0.60) KDM4EMTNR1AMTNR1BKMT2AMAOA
SCHEMBL14028586 0.86 PARP1 (0.58) KDM4EMTNR1AMTNR1BKMT2AMAOA
SCHEMBL27715458 0.80 PARP1 (0.76) MAOACYP1A2ADRA2ASLC6A2HTR2C
SCHEMBL10222677 0.80 BAZ2B (0.57) KDM4EMTNR1AMTNR1BKMT2AMAOA
SCHEMBL6070648 0.79 MAPK10 (0.55) KDM4EMTNR1AMTNR1BKMT2AMAOA
SCHEMBL30251048 0.76 CA1 (0.69) KDM4EKMT2ACA1CA2CA4
SCHEMBL4627835 0.76 CA1 (0.69) KDM4EKMT2ACA1CA2CA4
SCHEMBL7722965 0.76 MTNR1A (1.00) KDM4EMTNR1AMTNR1BKMT2AMAOA
SCHEMBL31488126 0.76 MTNR1A (1.00) KDM4EMTNR1AMTNR1BKMT2AMAOA
SCHEMBL8946440 0.76 CA1 (0.63) CA1CA2CA4CA6CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5185360-A Antioxidants, free radical scavengers UNIVERSITY OF BATH (GB) 1993-02-09 US disclosed
WO-1990015800-A1 INDENOINDOLE COMPOUNDS UNIVERSITY OF BATH (GB) 1990-12-27 WO disclosed
EP-0404536-A1 Indenoindole compounds I UNIVERSITY OF BATH (GB) 1990-12-27 EP disclosed