SCHEMBL9527334

SCHEMBL9527334

Cc1cccnc1C[S+]([O-])c1nc2cc(OC(F)(F)F)ccc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 3/20 0.40
RUNX1 Q01196 6/20 0.40
IDO1 P14902 1/20 0.35
PDE10A Q9Y233 1/20 0.34
KIT P10721 1/20 0.34
IDH1 O75874 2/20 0.33
CETP P11597 1/20 0.33
SLC40A1 Q9NP59 1/20 0.33
PDE2A O00408 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527662 0.92 RUNX1 (0.33) CBFBRUNX1
SCHEMBL9527362 0.91 ATP4A (0.40) CBFBRUNX1PDE2ATRPV1
SCHEMBL9527256 0.91 CBFB (0.34) CBFBRUNX1
SCHEMBL9526251 0.89 ATP4A (0.38) PDE10ATRPV1
SCHEMBL9528109 0.88 CYP3A4 (0.40) CBFB
SCHEMBL9526905 0.86 CBFB (0.35) CBFBRUNX1PDE10ATRPV1PTGS1
SCHEMBL10713063 0.85 KIF11 (0.39) CBFBPDE10APDE2ATRPV1
SCHEMBL23988513 0.83 ATP4A (0.45) CBFBRUNX1
SCHEMBL9527817 0.83 ATP4A (0.36) CBFBRUNX1PDE10A
SCHEMBL9527017 0.83 ATP4A (0.45) CBFBRUNX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0134400-B1 FLUOROALKOXYSUBSTITUTED PYRIDYLMETHYLTHIO-(OR SULFINYL-)BENZIMIDAZOLES HAVING A SECRETOLYTIC ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1993-03-24 EP disclosed
US-4555518-A ANTIULCER AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1985-11-26 US disclosed
EP-0134400-A2 Fluoroalkoxysubstituted pyridylmethylthio-(or sulfinyl-)benzimidazoles having a secretolytic activity Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1985-03-20 EP disclosed