SCHEMBL9528448

SCHEMBL9528448

CC(=O)C(C)(C)Cc1cccc(C)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.45
CTBP2 P56545 1/20 0.45
POLB P06746 1/20 0.44
ACHE P22303 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 1/20 0.42
RECQL P46063 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
IDO1 P14902 2/20 0.42
HPGD P15428 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MMP13 P45452 1/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.41
BRD4 O60885 1/20 0.40
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21859555 0.86 TAAR1 (0.47) MAOBCTBP2POLBACHETAAR1
SCHEMBL692554 0.86 CTBP2 (0.49) MAOBCTBP2POLBACHETAAR1
SCHEMBL17106362 0.81 MAOB (0.42) MAOBCTBP2POLBKDM4EALDH1A1
SCHEMBL20859039 0.81 CTBP2 (0.45) MAOBCTBP2POLBACHETAAR1
SCHEMBL10478213 0.81 TAAR1 (0.40) MAOBCTBP2POLBACHETAAR1
SCHEMBL12913271 0.81 RIPK1 (0.52) MAOBTAAR1KDM4E
SCHEMBL19047449 0.80 POLB (0.43) MAOBCTBP2POLBACHETAAR1
SCHEMBL19006263 0.80 MMP8 (0.48) MAOBCTBP2POLBALDH1A1RECQL
SCHEMBL20715896 0.79 ATM (0.37) CTBP2POLBKDM4EALDH1A1CYP3A4
SCHEMBL6552350 0.79 SMN1; SMN2 (0.50) TAAR1ALDH1A1CYP3A4RECQLLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017112617-A1 4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES MERCK SHARP & DOHME CORP. (US) 2017-06-29 WO disclosed
EP-0289913-B1 PARASITICIDAL AGENT BASED ON SUBSTITUTED AMINOMETHYL HETEROCYCLES BAYER AG (DE) 1993-01-13 EP disclosed
US-5128368-A Fungicides, bactericides BAYER AKTIENGESELLSCHAFT (DE) 1992-07-07 US disclosed
US-4988729-A 1,3-Dioxolane fungicides, bactericides applied to the habitat BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
EP-0256367-B1 SUBSTITUTED HYDROXY PROPYLAMINE DERIVATIVES BAYER AG (DE) 1990-08-29 EP disclosed
US-4845098-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-07-04 US disclosed
EP-0289913-A2 Parasiticidal agent based on substituted aminomethyl heterocycles BAYER AG (DE) 1988-11-09 EP disclosed
EP-0256367-A1 Substituted hydroxy propylamine derivatives BAYER AG (DE) 1988-02-24 EP disclosed