SCHEMBL9528889

SCHEMBL9528889

CCC[n+]1cc(Br)cc(C(=O)N(CCC(=O)NCCOC(=O)C2NCCc3ccccc32)c2ccccc2)c1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
OPRM1 P35372 6/20 0.32
OPRK1 P41145 4/20 0.32
ROCK2 O75116 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC18A2 Q05940 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9523922 0.99 TSHR (0.33) TSHRNPSR1OPRM1OPRK1ROCK2
SCHEMBL9525650 0.92 OPRM1 (0.34) TSHRNPSR1OPRM1OPRK1ROCK2
Hydrochloric Acid SCHEMBL9524987 0.92 OPRM1 (0.34) TSHRNPSR1OPRM1OPRK1ROCK2
Hydrochloric Acid SCHEMBL9523744 0.92 OPRM1 (0.34) TSHRNPSR1OPRM1OPRK1ROCK2
Hydrochloric Acid SCHEMBL9525305 0.91 TSHR (0.33) TSHRNPSR1OPRM1OPRK1ROCK2
Hydrochloric Acid SCHEMBL9525481 0.88 SLC18A2 (0.31) TSHRNPSR1SLC18A2
SCHEMBL9524781 0.85 NPC1 (0.38) TSHRNPSR1OPRM1ROCK2SLC6A2
Hydrochloric Acid SCHEMBL9528597 0.84 TSHR (0.39) TSHRNPSR1OPRM1OPRK1ROCK2
Hydrochloric Acid SCHEMBL9525523 0.83 THRA (0.36) TSHRNPSR1OPRM1OPRK1ROCK2
Hydrochloric Acid SCHEMBL9525127 0.82 TSHR (0.31) TSHRNPSR1OPRM1OPRK1SLC18A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP claimed
EP-0369810-A2 PAF antagonists as anti-hyperendothelinemia agents Takeda Chemical Industries, Ltd. (JP) 1990-05-23 EP claimed