SCHEMBL9529268

SCHEMBL9529268

CS(=O)(=O)Nc1cccc([C@@H](N)C([NH])=O)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
POLB P06746 1/20 0.50
KEAP1 Q14145 1/20 0.44
HPGD P15428 1/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
KIF11 P52732 1/20 0.40
DHX9 Q08211 1/20 0.40
CA2 P00918 1/20 0.40
KDM1A O60341 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10332567 1.00 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2POLBKEAP1HPGD
SCHEMBL8120763 0.87 HPGD (0.41) ALDH1A1SMN1; SMN2HPGDCA2ADRA1A
SCHEMBL11466281 0.86 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2POLBKEAP1HPGD
SCHEMBL8867750 0.86 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2POLBKEAP1HPGD
SCHEMBL8867745 0.86 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2POLBKEAP1HPGD
SCHEMBL11653449 0.84 POLB (0.56) ALDH1A1SMN1; SMN2POLBKEAP1HPGD
SCHEMBL4370199 0.79 KEAP1 (0.52) ALDH1A1SMN1; SMN2POLBKEAP1HSD17B1
SCHEMBL28012269 0.76 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2POLBKEAP1HPGD
SCHEMBL245468 0.76 MEN1 (0.60) ALDH1A1SMN1; SMN2POLBKEAP1HSD17B1
SCHEMBL10100499 0.75 KEAP1 (0.55) ALDH1A1SMN1; SMN2POLBKEAP1HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0187500-B1 MONOBACTAMS THE UPJOHN COMPANY (US) 1993-04-28 EP disclosed
EP-0187500-A1 Monobactams THE UPJOHN COMPANY (US) 1986-07-16 EP disclosed