SCHEMBL9529319

SCHEMBL9529319

CC(=O)Oc1cccc2c1CCN(C(=O)Cc1ccc(Cl)c(Cl)c1)C2CN1CCCC1

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 11/20 0.75
OPRK1 P41145 7/20 0.75
NPC1 O15118 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
NFKB1 P19838 1/20 0.51
CYP2C19 P33261 1/20 0.51
HIF1A Q16665 1/20 0.51
TDP1 Q9NUW8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9531087 0.99 OPRD1 (0.76) OPRD1OPRK1NPC1
SCHEMBL7642832 0.91 OPRD1 (0.75) OPRD1OPRK1NPC1CYP1A2CYP3A4
SCHEMBL9528558 0.91 OPRD1 (0.78) OPRD1OPRK1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9532360 0.90 OPRD1 (0.77) OPRD1OPRK1
SCHEMBL9529598 0.87 OPRD1 (0.87) OPRD1OPRK1NPC1CYP1A2CYP3A4
Fumaric Acid SCHEMBL10516264 0.86 OPRD1 (0.71) OPRD1OPRK1CYP3A4CYP2D6CYP2C9
Maleic Acid SCHEMBL10516259 0.86 OPRD1 (0.71) OPRD1OPRK1CYP3A4CYP2D6CYP2C9
SCHEMBL9528008 0.86 OPRD1 (0.82) OPRD1OPRK1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9528583 0.86 OPRD1 (0.87) OPRD1OPRK1NPC1
SCHEMBL9527997 0.86 OPRD1 (1.00) OPRD1OPRK1NPC1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0330360-B1 1,2,3,4-Tetrahydroisoquinolines, processes for their preparation, and their use as kappa-receptor agonists SMITHKLINE BEECHAM FARMA (IT) 1993-12-01 EP claimed