SCHEMBL9529417

SCHEMBL9529417

COc1ccc2c(c1)CCN(C(=O)Cc1ccc(Cl)c(Cl)c1)C2CN(C)C

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 5/20 0.64
OPRD1 P41143 6/20 0.63
TP53 P04637 1/20 0.49
MTNR1B P49286 1/20 0.48
GRIN2C Q14957 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9530248 0.99 OPRK1 (0.62) OPRK1OPRD1TP53MTNR1BGRIN2C
SCHEMBL9529566 0.93 OPRK1 (0.64) OPRK1OPRD1TP53MTNR1BPOLB
Hydrochloric Acid SCHEMBL9529311 0.92 OPRK1 (0.62) OPRK1OPRD1TP53MTNR1BPOLB
SCHEMBL9529202 0.88 OPRK1 (0.68) OPRK1OPRD1
SCHEMBL9528674 0.88 OPRD1 (0.70) OPRK1OPRD1
Hydrochloric Acid SCHEMBL9531229 0.87 OPRD1 (0.69) OPRK1OPRD1
SCHEMBL9529138 0.86 OPRD1 (0.73) OPRK1OPRD1
SCHEMBL9815269 0.85 OPRD1 (0.83) OPRK1OPRD1
Hydrochloric Acid SCHEMBL9529695 0.85 OPRD1 (0.72) OPRK1OPRD1
Hydrochloric Acid SCHEMBL9815302 0.84 OPRD1 (0.81) OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0330360-B1 1,2,3,4-Tetrahydroisoquinolines, processes for their preparation, and their use as kappa-receptor agonists SMITHKLINE BEECHAM FARMA (IT) 1993-12-01 EP claimed
EP-0330360-A1 1,2,3,4-Tetrahydroisoquinolines, processes for their preparation, and their use as kappa-receptor agonists SmithKline Beecham Farmaceutici S.p.A. (IT) 1989-08-30 EP claimed