SCHEMBL9529549

SCHEMBL9529549

CCOC(=O)c1cc2ccc3ccccc3c2o1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.54
ALDH1A1 P00352 5/20 0.54
GAA P10253 4/20 0.54
GLA P06280 1/20 0.54
KMT2A Q03164 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
MAPK1 P28482 2/20 0.51
MAPT P10636 6/20 0.50
NPC1 O15118 3/20 0.50
MEN1 O00255 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
RECQL P46063 1/20 0.50
CDC25B P30305 3/20 0.49
RAB9A P51151 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
CASP3 P42574 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537147 0.93 KDM4E (0.54) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL9540661 0.91 KDM4E (0.51) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL9778968 0.87 GAA (0.46) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL5311626 0.82 MAOA (0.53) KDM4EALDH1A1KMT2AMAPK1MAPT
SCHEMBL4675984 0.82 MAOA (0.68) KDM4EALDH1A1GAAKMT2AMAPK1
SCHEMBL11144122 0.82 MAOB (0.72) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL16271258 0.82 KDM4E (0.70) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL7469464 0.81 MAOB (0.52) KDM4EALDH1A1KMT2AMAPK1MAPT
SCHEMBL28805121 0.81 ALDH1A1 (0.59) KDM4EALDH1A1GAAGLAKMT2A
SCHEMBL931020 0.80 MAOB (0.51) KDM4EALDH1A1KMT2AMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4965285-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-10-23 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed