SCHEMBL9532585

SCHEMBL9532585

CC(=O)c1cccc(NC(=O)C2CCC2)c1

nearest known ligand 0.94

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.91
NPSR1 Q6W5P4 1/20 0.66
GAA P10253 2/20 0.64
KCNK3 O14649 1/20 0.63
KCNK9 Q9NPC2 1/20 0.63
TP53 P04637 1/20 0.62
USP2 O75604 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
NPC1 O15118 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
PKM P14618 1/20 0.59
ALOX15 P16050 1/20 0.59
LMNA P02545 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18664786 0.95 ALDH1A1 (1.00) ALDH1A1NPSR1GAAKCNK3KCNK9
SCHEMBL5816312 0.94 ALDH1A1 (0.85) ALDH1A1NPSR1GAAKCNK3KCNK9
SCHEMBL8352882 0.84 ALDH1A1 (0.71) ALDH1A1GAATP53USP2NPC1
SCHEMBL2892842 0.84 ALDH1A1 (0.71) ALDH1A1GAATP53USP2
SCHEMBL23070448 0.83 ALDH1A1 (0.78) ALDH1A1NPSR1GAAKCNK3KCNK9
SCHEMBL12764072 0.83 NPSR1 (0.94) ALDH1A1NPSR1GAAUSP2SMN1; SMN2
SCHEMBL16670220 0.82 ALDH1A1 (0.77) ALDH1A1NPSR1GAAKCNK3KCNK9
SCHEMBL13370008 0.81 ALDH1A1 (0.74) ALDH1A1NPSR1GAAKCNK3KCNK9
SCHEMBL12825257 0.81 NPSR1 (0.65) ALDH1A1NPSR1GAAKCNK3KCNK9
SCHEMBL20608480 0.81 GAA (0.77) ALDH1A1NPSR1GAAKCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0208846-B1 [7-(3-Disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID CO (US) 1993-11-18 EP disclosed
US-4654347-A USEFUL AS ANXIOLYTIC AND ANTIEPILEPTIC AGENTS, SEDATIVE-HYPNOTIC AGENTS AND SKELETAL MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1987-03-31 US disclosed
EP-0208846-A1 [7-(3-Disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1987-01-21 EP disclosed
US-4626538-A [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1986-12-02 US disclosed