SCHEMBL9533189

SCHEMBL9533189

CCCN(CCNS(C)(=O)=O)C1Cc2c[nH]c3ccc(OC)c(c23)C1

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.55
HTR1D P28221 8/20 0.50
HTR1B P28222 7/20 0.50
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
DRD2 P14416 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9776420 0.94 HTR1A (0.53) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL6890172 0.88 HTR1A (0.65) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL9534913 0.88 HTR1A (0.50) HTR1AHTR1DHTR1BMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7716614 0.87 HTR1A (0.64) HTR1AHTR1DHTR1BMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL9776382 0.87 HTR1A (0.49) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL10340387 0.84 HTR1A (0.60) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL9534014 0.84 HTR1A (0.56) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL9531561 0.83 HTR1A (0.59) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL9536727 0.83 HTR1A (0.57) HTR1AHTR1DHTR1BMTNR1AMTNR1B
SCHEMBL9776435 0.82 HTR1D (0.44) HTR1AHTR1DHTR1BMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021438-A Having affinity for 5-hydroxytryptamine receptors; treating central nervous system and cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1991-06-04 US claimed
EP-0332968-B1 1,3,4,5-Tetrahydrobenz[c,d]indoles BAYER AG (DE) 1993-06-02 EP disclosed
US-5021438-A Having affinity for 5-hydroxytryptamine receptors; treating central nervous system and cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1991-06-04 US disclosed
EP-0332968-A1 1,3,4,5-Tetrahydrobenz[c,d]indoles BAYER AG (DE) 1989-09-20 EP disclosed