SCHEMBL9533960

SCHEMBL9533960

CC(C#N)c1oc2ccc(Cl)c3c2c1CN(C)CC3

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 6/20 0.60
ADRA2B P18089 5/20 0.60
ADRA2C P18825 5/20 0.60
ADRA1A P35348 5/20 0.60
ADRA1D P25100 4/20 0.60
ADRA1B P35368 4/20 0.60
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CYP2D6 P10635 2/20 0.35
NPSR1 Q6W5P4 1/20 0.34
CYP1A2 P05177 1/20 0.32
HTR6 P50406 2/20 0.31
CHRM2 P08172 1/20 0.30
HTR1A P08908 1/20 0.30
CHRM1 P11229 1/20 0.30
DRD1 P21728 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378219 0.84 ADRA2A (0.64) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9535723 0.81 ADRA2A (0.60) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9382518 0.80 ADRA2A (0.65) ADRA2AADRA2BADRA2CADRA1AADRA1D
Hydrochloric Acid SCHEMBL9380664 0.79 ADRA2A (0.64) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9379201 0.77 ADRA2A (0.74) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9380112 0.77 ADRA2A (0.61) ADRA2AADRA2BADRA2CADRA1AADRA1D
Hydrochloric Acid SCHEMBL9380197 0.76 ADRA2A (0.72) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9380851 0.76 ADRA2A (0.72) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9380764 0.76 ADRA2A (0.60) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9383927 0.75 ADRA2A (0.62) ADRA2AADRA2BADRA2CADRA1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0384676-B1 Alpha-adrenergic receptor antagonists SMITHKLINE BEECHAM CORP (US) 1993-11-10 EP disclosed
US-4981849-A OBESITY, DIABETES, CARDIOVASCULAR DISORDERS, DEPRESSION SMITHKLINE BEECHAM CORPORATION (US) 1991-01-01 US disclosed
EP-0384676-A1 Alpha-adrenergic receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 1990-08-29 EP disclosed