SCHEMBL9534028

SCHEMBL9534028

O=C1NCCC12CC(COCc1ccccc1)Oc1ccc(F)cc12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.45
AKR1B1 P15121 9/20 0.43
BACE1 P56817 1/20 0.38
AKR1B10 O60218 1/20 0.35
AKR1A1 P14550 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
HRH4 Q9H3N8 4/20 0.33
HRH3 Q9Y5N1 4/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9432478 0.70 AKR1B1 (0.53) AKR1B1OPRM1OPRD1OPRK1
SCHEMBL9432167 0.66 AKR1B1 (0.44) AKR1B1OPRM1OPRD1OPRK1
SCHEMBL9432976 0.64 AKR1B1 (0.47) AKR1B1OPRM1OPRD1OPRK1
SCHEMBL5708359 0.63 LMNA (1.00) LMNAL3MBTL1HRH4HRH3
SCHEMBL1269358 0.63 LMNA (1.00) LMNAL3MBTL1HRH4HRH3
SCHEMBL18844035 0.63 LMNA (1.00) LMNAL3MBTL1HRH4HRH3
SCHEMBL3142790 0.62 LMNA (0.63) LMNAL3MBTL1HRH4HRH3
SCHEMBL10120126 0.61 LMNA (0.51) LMNAL3MBTL1HRH4HRH3
SCHEMBL9257211 0.61 AKR1B1 (0.66) AKR1B1AKR1B10AKR1A1
SCHEMBL9774876 0.60 LMNA (0.50) LMNAL3MBTL1HRH4HRH3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530198-A1 HETEROCYCLIC COMPOUNDS AS ALDOSE REDUCTASE INHIBITORS PFIZER INC. (US) 1993-03-10 EP disclosed
WO-1991015491-A1 HETEROCYCLIC COMPOUNDS AS ALDOSE REDUCTASE INHIBITORS PFIZER INC. (US) 1991-10-17 WO disclosed