SCHEMBL9534675

SCHEMBL9534675

CC(C)c1onc(-c2ccc(Cl)cc2)c1OC(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 8/20 0.44
THRB P10828 1/20 0.43
GABRA5 P31644 5/20 0.40
FFAR4 Q5NUL3 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NR1H4 Q96RI1 2/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPK9 P45984 1/20 0.36
CSNK1D P48730 1/20 0.36
MAPK10 P53779 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9533383 0.82 GPBAR1 (0.51) GPBAR1GABRA5FFAR4
SCHEMBL9535597 0.80 NR1H4 (0.53) NR1H4
SCHEMBL9535705 0.78 GPBAR1 (0.48) GPBAR1GABRA5FFAR4SMN1; SMN2
SCHEMBL9535545 0.76 FFAR4 (0.50) GPBAR1GABRA5FFAR4SMN1; SMN2
SCHEMBL9533125 0.75 KMT2A (0.48) GPBAR1SMN1; SMN2NR1H4ALDH1A1
SCHEMBL9535701 0.69 KMT2A (0.54) GPBAR1SMN1; SMN2
SCHEMBL29142635 0.68 GABRA5 (0.50) GPBAR1THRBGABRA5SMN1; SMN2ALDH1A1
SCHEMBL29142636 0.68 GABRA5 (0.50) GPBAR1THRBGABRA5SMN1; SMN2ALDH1A1
SCHEMBL11519685 0.67 KMT2A (0.51) GPBAR1SMN1; SMN2NR1H4
SCHEMBL27565925 0.66 GPBAR1 (0.40) GPBAR1THRBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573883-A1 Utilization of 3 substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives against endoparasites new 3-substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives and process for their preparation BAYER AG (DE) 1993-12-15 EP disclosed