SCHEMBL9534898

SCHEMBL9534898

CCOC(=O)CC[C@H](NC(=O)c1ccc(CCC2CNc3nc(N)nc(N)c3C2)cc1)C(=O)OCC

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.58
GART P22102 3/20 0.56
ATIC P31939 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9534903 1.00 DHFR (0.58) DHFRGARTATIC
SCHEMBL9446065 0.95 DHFR (0.53) DHFRGART
SCHEMBL9383614 0.93 GART (0.56) DHFRGARTATIC
SCHEMBL9383606 0.93 GART (0.56) DHFRGARTATIC
SCHEMBL9446079 0.89 GART (0.51) DHFRGARTATIC
SCHEMBL9446085 0.89 GART (0.51) DHFRGARTATIC
SCHEMBL9536119 0.85 GART (0.77) DHFRGARTATIC
SCHEMBL9534086 0.84 GART (0.49) DHFRGARTATIC
SCHEMBL9534079 0.84 GART (0.49) DHFRGARTATIC
SCHEMBL9536782 0.84 GART (0.68) DHFRGARTATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4684653-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1987-08-04 US claimed
EP-0215063-B1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES UNIV PRINCETON (US) 1993-11-03 EP disclosed
US-5026851-A Antineoplastic agents THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-25 US disclosed
US-4845216-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-07-04 US disclosed
EP-0215063-A4 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES. UNIV PRINCETON (US) 1987-11-23 EP disclosed
US-4684653-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1987-08-04 US disclosed
EP-0215063-A1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES. UNIV PRINCETON (US) 1987-03-25 EP disclosed
WO-1986005181-A1 PYRIDO AD2,3-d BDPYRIMIDIN DERIVATIVES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1986-09-12 WO disclosed