SCHEMBL9534949

SCHEMBL9534949

CC(CC1CNc2nc(N)nc(O)c2C1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GART P22102 6/20 0.58
ATIC P31939 3/20 0.52
DHFR P00374 1/20 0.49
SOST Q9BQB4 1/20 0.46
MTHFD2 P13995 2/20 0.46
MTHFD1 P11586 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535744 0.94 GART (0.51) GARTATICDHFRSOST
SCHEMBL9446048 0.93 GART (0.61) GARTATICDHFRSOSTMTHFD1
SCHEMBL9535135 0.93 GART (0.58) GARTATICDHFR
SCHEMBL9536040 0.91 GART (0.56) GARTATICDHFR
SCHEMBL10479205 0.90 GART (0.57) GARTATICSOSTMTHFD2MTHFD1
SCHEMBL10479151 0.90 GART (0.57) GARTATICSOSTMTHFD2MTHFD1
SCHEMBL10479154 0.90 GART (0.57) GARTATICSOSTMTHFD2MTHFD1
SCHEMBL10479169 0.90 GART (0.57) GARTATICSOSTMTHFD2MTHFD1
SCHEMBL10479203 0.90 GART (0.57) GARTATICSOSTMTHFD2MTHFD1
SCHEMBL9535149 0.87 GART (0.52) GARTATICDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215063-B1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES UNIV PRINCETON (US) 1993-11-03 EP claimed
US-4684653-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1987-08-04 US claimed
US-4845216-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-07-04 US disclosed
US-4684653-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1987-08-04 US disclosed