SCHEMBL9534952

SCHEMBL9534952

CN(C)CCn1c(NC2CCNCC2)nc2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.61
NR4A2 P43354 1/20 0.61
POLB P06746 1/20 0.56
KDM4E B2RXH2 2/20 0.49
HIF1A Q16665 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
LMNA P02545 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
SSTR5 P35346 2/20 0.43
RPS6KA2 Q15349 1/20 0.43
TOP2A P11388 1/20 0.43
TP53 P04637 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
RECQL P46063 1/20 0.43
BLM P54132 1/20 0.43
HBB P68871 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7985049 0.84 KCNH2 (0.65) KCNH2NR4A2SSTR5
SCHEMBL6991613 0.82 KCNH2 (0.59) KCNH2NR4A2KDM4EALDH1A1
SCHEMBL7981124 0.81 KCNH2 (0.61) KCNH2NR4A2POLBCYP1A2CYP3A4
SCHEMBL6992893 0.81 KCNH2 (0.59) KCNH2NR4A2KDM4EALDH1A1LMNA
SCHEMBL7980989 0.81 KCNH2 (0.58) KCNH2NR4A2KDM4EALDH1A1LMNA
SCHEMBL5537223 0.81 KCNH2 (0.58) KCNH2NR4A2LMNACYP1A2CYP3A4
SCHEMBL9535562 0.81 KCNH2 (0.60) KCNH2NR4A2ALDH1A1HPGDLMNA
SCHEMBL13319057 0.81 KCNH2 (0.63) KCNH2NR4A2HIF1AALDH1A1HPGD
SCHEMBL6991720 0.80 KCNH2 (0.57) KCNH2NR4A2POLBKDM4EHIF1A
Hydrochloric Acid SCHEMBL5009615 0.80 KCNH2 (0.58) KCNH2NR4A2KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0282133-B1 1-ALKYL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-07-28 EP disclosed
EP-0282133-A2 1-alkyl substituted benzimidazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-09-14 EP disclosed