SCHEMBL9535289

SCHEMBL9535289

Cc1ccc(Cc2cccc(N)c2N)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.48
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 2/20 0.38
CYP3A4 P08684 2/20 0.38
PIK3CA P42336 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2A6 P11509 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
LTA4H P09960 2/20 0.37
AGXT P21549 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10610547 0.84 CYP3A4 (0.52) CD44ALDH1A1TSHRCYP3A4TDP1
SCHEMBL11658684 0.84 POLB (0.44) POLBKDM4EALDH1A1HPGDTSHR
SCHEMBL28680564 0.83 KCNH2 (0.46) CD44KDM4EALDH1A1HPGDTSHR
SCHEMBL102570 0.82 HTR2A (0.50) CD44POLBHPGDCYP3A4CYP1A2
SCHEMBL2776883 0.81 MEN1 (0.41) CD44ALDH1A1HPGDCYP3A4TAAR1
Nitrogen SCHEMBL27535571 0.81 POLB (0.41) POLBKDM4EALDH1A1HPGDTSHR
SCHEMBL27535570 0.79 LTA4H (0.33) POLBTSHRCYP1A2CYP2A6TAAR1
SCHEMBL5793478 0.79 POLB (0.43) POLBKDM4EALDH1A1HPGDTSHR
SCHEMBL3132841 0.79 CD44 (0.46) CD44POLBALDH1A1HPGDTSHR
SCHEMBL6648051 0.77 LOXL2 (0.45) CD44CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed