SCHEMBL9535658

SCHEMBL9535658

[CH2]C(SC)c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.44
TSHR P16473 2/20 0.41
MAPK1 P28482 2/20 0.41
HIF1A Q16665 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
AOC3 Q16853 1/20 0.38
CYP2A6 P11509 1/20 0.38
BRD4 O60885 1/20 0.38
CYP19A1 P11511 3/20 0.37
IDO1 P14902 2/20 0.37
TDO2 P48775 2/20 0.37
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 3/20 0.36
SLC6A2 P23975 1/20 0.34
FFAR2 O15552 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8802618 0.78 CHRNA7 (0.41) TDP1CYP19A1
SCHEMBL11572011 0.75 SLC6A4 (0.48) ADRB2TSHRMAPK1HIF1ATDP1
SCHEMBL6295188 0.75 DPP4 (0.38) TSHRHIF1ATDP1LMNA
SCHEMBL1145645 0.73 ADRB2 (0.52) ADRB2TSHRMAPK1HIF1ATDP1
SCHEMBL1003900 0.72 ADRB2 (0.56) ADRB2TSHRMAPK1HIF1ATDP1
SCHEMBL3754314 0.72 ADRB2 (0.56) ADRB2TSHRMAPK1HIF1ATDP1
SCHEMBL3745333 0.72 ADRB2 (0.56) ADRB2TSHRMAPK1HIF1ATDP1
SCHEMBL8041464 0.71 CYP3A4 (0.43) TSHRMAPK1LMNACYP19A1SLC6A4
SCHEMBL3535353 0.71 TSHR (0.50) ADRB2TSHRMAPK1HIF1ATDP1
SCHEMBL25304239 0.70 ADRB2 (0.54) ADRB2TSHRMAPK1HIF1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0347146-B1 FUSED PYRIMIDINE DERIVATIVES, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-09-01 EP claimed