SCHEMBL9535689

SCHEMBL9535689

CNC1CCC2=C1CN(c1cc3c(cc1F)c(=O)c(C(=O)O)cn3C(C)(C)C)C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.44
KDM4E B2RXH2 9/20 0.44
LMNA P02545 7/20 0.43
HPGD P15428 6/20 0.43
HSD17B10 Q99714 6/20 0.43
MAPT P10636 1/20 0.43
CYP1A2 P05177 1/20 0.43
TOP2A P11388 1/20 0.43
CYP2C9 P11712 1/20 0.43
TOP2B Q02880 1/20 0.43
TOP1 P11387 1/20 0.42
DRD3 P35462 1/20 0.42
HTT P42858 3/20 0.41
TSHR P16473 2/20 0.41
BRD4 O60885 1/20 0.41
CYP2J2 P51589 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535816 0.88 ALDH1A1 (0.45) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9535484 0.86 DRD3 (0.59) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9538815 0.84 KDM4E (0.42) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9534436 0.82 ALDH1A1 (0.44) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9147720 0.76 ALDH1A1 (0.49) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9685920 0.76 ALDH1A1 (0.54) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9686875 0.75 ALDH1A1 (0.73) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9685571 0.75 ALDH1A1 (0.61) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9045127 0.75 TOP1 (0.61) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9686810 0.75 ALDH1A1 (0.50) ALDH1A1KDM4ELMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549857-A1 Antibacterial quinolone carboxylic acid derivatives KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1993-07-07 EP disclosed
EP-0550019-A2 Novel quinolone carboxylic acid derivatives and processes for preparing same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1993-07-07 EP disclosed