SCHEMBL9686875

SCHEMBL9686875

CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)cn3C(C)(C)C)CC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.73
DRD3 P35462 1/20 0.70
LMNA P02545 4/20 0.66
MEN1 O00255 3/20 0.66
KMT2A Q03164 3/20 0.66
KDM4E B2RXH2 9/20 0.64
HPGD P15428 4/20 0.64
NPC1 O15118 1/20 0.64
HSD17B10 Q99714 4/20 0.55
GAA P10253 1/20 0.55
RAD52 P43351 1/20 0.55
BRD4 O60885 1/20 0.54
TSHR P16473 1/20 0.54
HTT P42858 1/20 0.54
CYP2J2 P51589 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
MAPT P10636 1/20 0.54
CYP1A2 P05177 1/20 0.52
TOP2A P11388 1/20 0.52
CYP2C9 P11712 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685571 0.91 ALDH1A1 (0.61) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9685705 0.88 ALDH1A1 (0.58) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9685706 0.88 ALDH1A1 (0.70) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL11394177 0.86 ALDH1A1 (0.76) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL29388444 0.84 ALDH1A1 (1.00) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL7809357 0.84 ALDH1A1 (1.00) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL10923356 0.84 ALDH1A1 (0.72) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9685920 0.83 ALDH1A1 (0.54) ALDH1A1DRD3LMNAMEN1KMT2A
SCHEMBL9686268 0.82 ALDH1A1 (0.52) ALDH1A1DRD3LMNAMEN1KMT2A
Pefloxacin SCHEMBL34292 0.82 DRD3 (1.00) ALDH1A1DRD3LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288519-A4 1-TERTIARY-ALKYL-SUBSTITUTED NAPHTHYRIDINE- AND QUINOLINE-CARBOXYLIC ACID ANTIBACTERIAL AGENTS 1992-04-15 EP disclosed
US-4965273-A Certain 1-tertiary-butyl-naphthyridone carboxylic acid derivatives anti-bacterial agents BRISTOL-MYERS COMPANY (US) 1990-10-23 US disclosed
US-4954507-A 1-tertiary-alkyl-substituted naphthyridine carboxylic acid antibacterial agents BRISTOL-MYERS COMPANY (US) 1990-09-04 US disclosed
EP-0288519-A1 1-TERTIARY-ALKYL-SUBSTITUTED NAPHTHYRIDINE- AND QUINOLINE-CARBOXYLIC ACID ANTIBACTERIAL AGENTS Bristol-Myers Squibb Company (US) 1988-11-02 EP disclosed
EP-0266576-A2 1-Tert-alkyl-substituted naphthyridine and quinoline carboxylic acids as antibacterial agents Bristol-Myers Squibb Company (US) 1988-05-11 EP disclosed
WO-1988002627-A1 1-TERTIARY-ALKYL-SUBSTITUTED NAPHTHYRIDINE- AND QUINOLINE-CARBOXYLIC ACID ANTIBACTERIAL AGENTS BRISTOL-MYERS COMPANY (US) 1988-04-21 WO disclosed