SCHEMBL9535823

SCHEMBL9535823

Cc1cc(=O)[nH]c(=O)n1C=CC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYMP P19971 15/20 0.45
ATM Q13315 1/20 0.36
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535833 0.77 SMN1; SMN2 (0.37) TYMPALDH1A1NPC1KDM4EGAA
SCHEMBL10786702 0.77 SMN1; SMN2 (0.37) TYMPALDH1A1NPC1KDM4EGAA
SCHEMBL19348252 0.67 CRBN (0.43) ATMALDH1A1KDM4EMEN1KMT2A
SCHEMBL4889955 0.66 TYMP (0.47) TYMPATMALDH1A1KDM4EMEN1
SCHEMBL6027678 0.65 TYMP (0.46) TYMPATMALDH1A1KDM4EGAA
SCHEMBL8768819 0.62 TYMP (0.44) TYMPATMALDH1A1KDM4EMEN1
SCHEMBL10565144 0.61 TYMP (0.40) TYMPATMALDH1A1KDM4EGAA
SCHEMBL18072360 0.60 HSD17B10 (0.53) TYMPATMALDH1A1KDM4EMEN1
SCHEMBL15469004 0.60 POLB (0.43) TYMPATMALDH1A1KDM4EGAA
SCHEMBL4960409 0.60 POLB (0.46) TYMPATMALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0168813-B1 Sparsomycin derivatives MERRELL DOW PHARMA (US) 1993-11-10 EP disclosed
EP-0108455-B1 SPARSOMYCIN (SC-RS) DERIVATIVE; PHARMACEUTICAL COMPOSITION HAVING ANTI-TUMOR ACTIVITY Stichting Katholieke Universiteit (NL) 1987-04-22 EP disclosed
US-4581360-A Sparsomycin (Sc -Rs) derivative; pharmaceutical composition having anti-tumor activity STICHTING KATHOLIEKE UNIVERSITEIT (NL) 1986-04-08 US disclosed
EP-0168813-A1 Sparsomycin derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1986-01-22 EP disclosed
EP-0108455-A1 Sparsomycin (Sc-Rs) derivative; pharmaceutical composition having anti-tumor activity Stichting Katholieke Universiteit (NL) 1984-05-16 EP disclosed