SCHEMBL9536296

SCHEMBL9536296

c1csc(NCCN2CCCCC2)n1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.46
MAPT P10636 1/20 0.42
LTA4H P09960 1/20 0.41
HRH1 P35367 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31084647 0.87 MAPT (0.45) MAPTHRH1SIGMAR1ALDH1A1TSHR
SCHEMBL23647320 0.84 CASR (0.46) MAPTALDH1A1TSHR
SCHEMBL6312404 0.79 ACHE (0.47) MAPTHRH1ALDH1A1
SCHEMBL11319195 0.79 SMN1; SMN2 (0.54) MAPTHRH1ALDH1A1TSHR
SCHEMBL11306755 0.77 SMN1; SMN2 (0.55) MAPTHRH1ALDH1A1TSHR
Hydrochloric Acid SCHEMBL7534025 0.74 SMN1; SMN2 (0.49) HRH3HRH1ALDH1A1
SCHEMBL9672230 0.73 HRH3 (0.54) HRH3SIGMAR1ALDH1A1
SCHEMBL9536249 0.72 KDM4E (0.53) ALDH1A1
SCHEMBL12894447 0.72 PLAU (0.46)
SCHEMBL29180050 0.70 ALDH1A1 (0.43) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
EP-0533781-A1 3-ARYL-2-HYDROXYPROPIONIC ACID DERIVATIVES AND ANALOGS AS HYPOGLYCEMIC AGENTS. PFIZER (US) 1993-03-31 EP disclosed