SCHEMBL9536685

SCHEMBL9536685

CCOC(=O)C1=C(CN=C(N)S)NC(C)=C(C#N)C1C1CCC1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.49
TSHR P16473 2/20 0.49
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
NR3C2 P08235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9212110 0.99 NPSR1 (0.48) NPSR1TSHRALDH1A1POLBCYP1A2
Hydrochloric Acid SCHEMBL9214116 0.97 NPSR1 (0.51) NPSR1TSHRALDH1A1POLBCYP1A2
Hydrochloric Acid SCHEMBL9212505 0.96 NPSR1 (0.53) NPSR1TSHRALDH1A1POLBCYP1A2
Hydrochloric Acid SCHEMBL9208633 0.96 NPSR1 (0.53) NPSR1TSHRALDH1A1POLBCYP1A2
SCHEMBL9211438 0.96 NPSR1 (0.46) NPSR1TSHRALDH1A1POLBCYP1A2
Hydrochloric Acid SCHEMBL9210456 0.95 NPSR1 (0.45) NPSR1TSHRALDH1A1POLBCYP1A2
Hydrochloric Acid SCHEMBL9339531 0.95 NPSR1 (0.45) NPSR1TSHRALDH1A1POLBCYP1A2
Hydrochloric Acid SCHEMBL9205116 0.83 ADORA3 (0.40) NPSR1TSHRALDH1A1POLBCYP1A2
SCHEMBL9203548 0.81 ADORA3 (0.40) NPSR1TSHRALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9212238 0.81 ADORA3 (0.40) NPSR1TSHRALDH1A1POLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536169-A1 3H,7H]THIAZOLO 3,4-a]PYRIDINES WITH ANTIASTHMATIC AND ANTIINFLAMMATORY ACTIONS ON THE RESPIRATORY TRACT. BOEHRINGER MANNHEIM ITALIA (IT) 1993-04-14 EP disclosed