SCHEMBL9536711

SCHEMBL9536711

Cc1nc2ccccn2c(=O)c1CCN1CCC(Cc2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.59
HTR1A P08908 3/20 0.59
HTR2C P28335 3/20 0.59
MEN1 O00255 2/20 0.59
CYP3A4 P08684 2/20 0.59
MAPT P10636 2/20 0.59
KMT2A Q03164 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
KDM4E B2RXH2 1/20 0.59
PKM P14618 1/20 0.59
HPGD P15428 1/20 0.59
TSHR P16473 1/20 0.59
THPO P40225 1/20 0.59
PMP22 Q01453 1/20 0.59
ACHE P22303 1/20 0.55
SSTR5 P35346 2/20 0.46
HRH1 P35367 5/20 0.45
TACR2 P21452 2/20 0.45
TACR1 P25103 2/20 0.45
KCNH2 Q12809 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10803117 0.91 HTR2C (0.56) CYP2D6HTR1AHTR2CMEN1CYP3A4
Bromide SCHEMBL10550913 0.90 HTR2C (0.56) CYP2D6HTR1AHTR2CMEN1CYP3A4
SCHEMBL9537351 0.90 HTR1A (0.56) CYP2D6HTR1AHTR2CMEN1CYP3A4
Oxalic Acid SCHEMBL10803137 0.89 HTR2C (0.55) CYP2D6HTR1AHTR2CMEN1CYP3A4
Oxalic Acid SCHEMBL10803132 0.89 HTR2C (0.55) CYP2D6HTR1AHTR2CMEN1CYP3A4
Hydrochloric Acid SCHEMBL9740582 0.88 CYP2D6 (0.56) CYP2D6HTR1AHTR2CMEN1CYP3A4
Oxalic Acid SCHEMBL10552172 0.86 HTR2C (0.54) CYP2D6HTR1AHTR2CMEN1CYP3A4
Oxalic Acid SCHEMBL10552180 0.86 HTR2C (0.54) CYP2D6HTR1AHTR2CMEN1CYP3A4
SCHEMBL9383006 0.86 SSTR5 (0.47) CYP2D6HTR1AHTR2CMEN1CYP3A4
SCHEMBL9536489 0.85 ADRA1A (0.48) CYP2D6HTR1AHTR2CMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed