SCHEMBL9537180

SCHEMBL9537180

CCn1c2ccccc2c2cc3ccccc3c(CNC(C)(CO)COS(C)(=O)=O)c21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.35
NPY5R Q15761 2/20 0.35
SLC2A1 P11166 1/20 0.35
MAPT P10636 5/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
LMNA P02545 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 2/20 0.33
POLB P06746 2/20 0.33
PTGER4 P35408 3/20 0.33
NPSR1 Q6W5P4 3/20 0.33
MAPK1 P28482 2/20 0.33
RAB9A P51151 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537186 0.90 SLC2A1 (0.42) RORCNPY5RSLC2A1MAPTMEN1
SCHEMBL9537938 0.87 NPY5R (0.39) NPY5RMAPTMEN1KMT2ALMNA
SCHEMBL9538345 0.84 RORC (0.38) RORCNPY5RSLC2A1MAPTMEN1
SCHEMBL10348691 0.81 SLC2A1 (0.39) SLC2A1KMT2ALMNACYP1A2CYP2D6
SCHEMBL9754641 0.80 SLC2A1 (0.45) RORCNPY5RSLC2A1MAPTMEN1
SCHEMBL10484383 0.79 SLC2A1 (0.40) SLC2A1MAPTKMT2ACYP1A2ALDH1A1
SCHEMBL10488353 0.78 SLC2A1 (0.37) SLC2A1MEN1KMT2A
SCHEMBL9538092 0.77 PER2 (0.35) NPY5RMAPTMEN1KMT2ALMNA
SCHEMBL9779025 0.76 SLC2A1 (0.36) SLC2A1KMT2ALMNACYP1A2CYP2C19
SCHEMBL9537789 0.76 SLC2A1 (0.42) SLC2A1MAPTKMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0182608-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-03-03 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed
EP-0182608-A2 Polycyclic compounds, their preparation and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-05-28 EP disclosed