SCHEMBL9537490

SCHEMBL9537490

Cc1c(C(=O)O)ncc2[nH]c3ccc(Oc4ccc([N+](=O)[O-])cc4)cc3c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
PKM P14618 1/20 0.46
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
GABRA1 P14867 8/20 0.44
GABRG2 P18507 8/20 0.44
GABRB3 P28472 8/20 0.44
GABRA5 P31644 8/20 0.44
GABRA2 P47869 8/20 0.44
GABRA3 P34903 7/20 0.44
KDM4E B2RXH2 2/20 0.44
GABRP O00591 4/20 0.43
GABRD O14764 4/20 0.43
GABRB1 P18505 4/20 0.43
GABRB2 P47870 4/20 0.43
GABRA4 P48169 4/20 0.43
GABRE P78334 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535854 0.88 GABRA1 (0.57) ALDH1A1MEN1KMT2AGABRA1GABRG2
SCHEMBL9533356 0.87 GABRA1 (0.51) ALDH1A1KMT2AGABRA1GABRG2GABRB3
SCHEMBL9537497 0.86 MEN1 (0.42) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL9535806 0.85 GABRA1 (0.57) ALDH1A1GABRA1GABRG2GABRB3GABRA5
SCHEMBL9536032 0.85 GABRA1 (0.47) ALDH1A1GABRA1GABRG2GABRB3GABRA5
SCHEMBL9538245 0.81 GABRA1 (0.44) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL9534871 0.81 MEN1 (0.48) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL9534774 0.80 GABRA1 (0.53) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL9537349 0.79 GABRA1 (0.74) ALDH1A1GABRA1GABRG2GABRB3GABRA5
SCHEMBL9535350 0.78 GABRA1 (0.56) ALDH1A1GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234173-B1 PHENOXY-SUBSTITUTED BETA-CARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 1993-06-16 EP disclosed
US-4945090-A ANXIOLYTIC AGENTS, ANTICONVULSANTS SCHERING AKTIENGESELLSCHAFT (DE) 1990-07-31 US disclosed
EP-0234173-A2 Phenoxy-substituted beta-carboline derivatives, their preparation and their use as medicaments SCHERING AKTIENGESELLSCHAFT (DE) 1987-09-02 EP disclosed