SCHEMBL9537754

SCHEMBL9537754

CCn1nnnc1SCCBr

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.79
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
POLB P06746 2/20 0.46
CYP2C19 P33261 2/20 0.43
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
TP53 P04637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
RCE1 Q9Y256 1/20 0.40
USP2 O75604 2/20 0.39
MAPT P10636 1/20 0.39
GAA P10253 1/20 0.39
GLA P06280 1/20 0.39
HTT P42858 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10971944 0.76 ALDH1A1 (0.69) ALDH1A1NPC1RAB9APOLBCYP2C19
SCHEMBL13814466 0.76 ALDH1A1 (0.69) ALDH1A1NPC1RAB9APOLBCYP2C19
SCHEMBL16072797 0.74 ALDH1A1 (0.67) ALDH1A1NPC1RAB9APOLBCYP2C19
SCHEMBL11069089 0.74
SCHEMBL9703552 0.72
SCHEMBL6897277 0.70 ALDH1A1 (0.61) ALDH1A1NPC1RAB9APOLBCYP2C19
SCHEMBL10671936 0.70 ALDH1A1 (0.58) ALDH1A1NPC1RAB9APOLBCYP2C19
SCHEMBL10675454 0.69 ALDH1A1 (0.56) ALDH1A1NPC1RAB9APOLBCYP2C19
SCHEMBL10969904 0.66 ALDH1A1 (0.58) ALDH1A1LMNASMN1; SMN2TP53GAA
SCHEMBL21916114 0.66 ALDH1A1 (0.59) ALDH1A1KMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed