SCHEMBL9538258

SCHEMBL9538258

CCOc1cc2cc(CO)sc2cc1OCC

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.44
STING1 Q86WV6 4/20 0.39
PTPN2 P17706 1/20 0.38
ALDH1A1 P00352 1/20 0.36
S1PR1 P21453 6/20 0.36
S1PR3 Q99500 3/20 0.36
TSHR P16473 2/20 0.36
CYP3A4 P08684 1/20 0.36
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 2/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33
GLA P06280 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541062 0.84 STING1 (0.36) STING1ALDH1A1S1PR1S1PR3TSHR
SCHEMBL9541014 0.83 ALDH1A1 (0.36) STING1ALDH1A1TSHRCYP3A4KMT2A
SCHEMBL7028472 0.82 PDE4A (0.50) CYP2A6STING1PTPN2
SCHEMBL9538537 0.81 STING1 (0.43) STING1ALDH1A1TSHRCYP3A4KMT2A
SCHEMBL9538461 0.79 STING1 (0.47) STING1TSHRCYP3A4HSD17B10TP53
SCHEMBL9537166 0.78 STING1 (0.33) STING1ALDH1A1TSHRKMT2AHSD17B10
SCHEMBL9541789 0.77 TSHR (0.40) STING1TSHRCYP3A4KMT2AHSD17B10
SCHEMBL10271885 0.77 KDM4E (0.39) STING1ALDH1A1TSHRCYP3A4KMT2A
SCHEMBL9540660 0.76 CYP3A4 (0.39) STING1TSHRCYP3A4
SCHEMBL9537019 0.73 STING1 (0.42) STING1ALDH1A1TSHRMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993005033-A1 BENZO[b]THIOPHENE DERIVATES, PROCESS FOR PRODUCING THE SAME AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1993-03-18 WO disclosed
US-4863923-A Method of inhibiting superoxide release ELI LILLY AND COMPANY (US) 1989-09-05 US disclosed
EP-0253650-A2 Improvements relating to benzothiophene derivatives ELI LILLY AND COMPANY (US) 1988-01-20 EP disclosed