SCHEMBL9541789

SCHEMBL9541789

CCOc1cc2cc(CN(O)C(C)=O)sc2cc1OCC

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
CYP3A4 P08684 1/20 0.40
STING1 Q86WV6 10/20 0.39
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CA9 Q16790 2/20 0.34
HSD17B10 Q99714 1/20 0.34
ALOX5 P09917 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539018 0.84 TSHR (0.36) TSHRCYP3A4STING1LMNATP53
SCHEMBL9538537 0.78 STING1 (0.43) TSHRCYP3A4STING1HSD17B10KMT2A
SCHEMBL9538258 0.77 CYP2A6 (0.44) TSHRCYP3A4STING1TP53HSD17B10
SCHEMBL9540660 0.77 CYP3A4 (0.39) TSHRCYP3A4STING1ALOX5
SCHEMBL9538461 0.76 STING1 (0.47) TSHRCYP3A4STING1TP53HSD17B10
SCHEMBL9541014 0.74 ALDH1A1 (0.36) TSHRCYP3A4STING1LMNAHSD17B10
SCHEMBL9541062 0.72 STING1 (0.36) TSHRCYP3A4STING1TP53HSD17B10
Tibenelast SCHEMBL449748 0.72 STING1 (0.54) TSHRSTING1HSD17B10
SCHEMBL9540466 0.71 PPARG (0.40) TSHRCYP3A4STING1
SCHEMBL9537019 0.71 STING1 (0.42) TSHRSTING1LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993005033-A1 BENZO[b]THIOPHENE DERIVATES, PROCESS FOR PRODUCING THE SAME AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1993-03-18 WO disclosed