SCHEMBL9538291

SCHEMBL9538291

N#Cc1ccc(-c2ccnc3ccccc23)[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 8/20 0.43
AURKA O14965 1/20 0.43
TTK P33981 1/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
BMPR1B O00238 2/20 0.43
BMPR1A P36894 2/20 0.43
ACVR1B P36896 2/20 0.43
ACVRL1 P37023 2/20 0.43
TGFBR1 P36897 2/20 0.43
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15074582 0.79 NPC1 (0.57) ACVR1AURKATTKAURKBINCENP
SCHEMBL9754547 0.77 MCL1 (0.55) KDM4EALDH1A1HPGDMDM2GLA
SCHEMBL29077121 0.76 ALDH1A1 (0.47) ACVR1NPC1RAB9AKDM4EALDH1A1
SCHEMBL7351074 0.74 AURKA (0.67) ACVR1AURKATTKAURKBINCENP
SCHEMBL9536884 0.73 KDM4E (0.46) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL11846505 0.73 KDM4E (0.49) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL9754396 0.72 ACVR1 (0.42) ACVR1AURKATTKAURKBINCENP
SCHEMBL9539748 0.71 FASN (0.46) KDM4EALDH1A1HPGDMDM2GLA
SCHEMBL3479396 0.71 KDM4E (0.53) KDM4EALDH1A1HPGDMDM2GLA
SCHEMBL15070838 0.71 GSK3B (0.61) ACVR1NPC1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532531-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-03-24 EP disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed