SCHEMBL9539965

SCHEMBL9539965

COCCc1ccc(OCC(O)CNC2CCCc3ccccc32)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.72
KDM4E B2RXH2 4/20 0.72
HTT P42858 2/20 0.66
ADRB1 P08588 4/20 0.62
KMT2A Q03164 3/20 0.62
ADRB2 P07550 3/20 0.62
MEN1 O00255 2/20 0.62
CYP1A2 P05177 2/20 0.62
TP53 P04637 1/20 0.62
CYP3A4 P08684 1/20 0.62
ADRB3 P13945 1/20 0.62
TSHR P16473 1/20 0.62
CYP2C19 P33261 1/20 0.62
CYP2D6 P10635 2/20 0.56
NR3C1 P04150 1/20 0.56
ADRA1A P35348 1/20 0.56
CYP2J2 P51589 1/20 0.56
PDE4D Q08499 1/20 0.56
LMNA P02545 3/20 0.56
TAAR1 Q96RJ0 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9589964 0.99 ALDH1A1 (0.71) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL14355265 0.86 KMT2A (0.69) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL9538697 0.83 ALDH1A1 (0.74) ALDH1A1KDM4EHTTADRB1KMT2A
Hydrochloric Acid SCHEMBL9586835 0.82 ALDH1A1 (0.72) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL9537291 0.81 ALDH1A1 (0.71) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL9539023 0.81 CYP2D6 (0.59) ALDH1A1KDM4EADRB1KMT2AADRB2
Hydrochloric Acid SCHEMBL9587817 0.81 ALDH1A1 (0.70) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL9540272 0.80 KMT2A (0.77) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL9588898 0.80 ALDH1A1 (0.90) ALDH1A1KDM4EHTTADRB1KMT2A
SCHEMBL9540740 0.80 ALDH1A1 (0.72) ALDH1A1KDM4EHTTADRB1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed