SCHEMBL9540740

SCHEMBL9540740

CC(=O)Nc1ccc(OCC(O)CNC2CCCc3ccccc32)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.72
HTT P42858 4/20 0.72
KDM4E B2RXH2 4/20 0.69
KMT2A Q03164 7/20 0.64
MEN1 O00255 4/20 0.64
TSHR P16473 3/20 0.64
CYP1A2 P05177 2/20 0.64
ADRB2 P07550 2/20 0.64
ADRB1 P08588 2/20 0.64
ADRB3 P13945 2/20 0.64
CYP2C19 P33261 2/20 0.64
TP53 P04637 1/20 0.64
CYP3A4 P08684 1/20 0.64
LMNA P02545 3/20 0.64
MAPT P10636 3/20 0.64
TAAR1 Q96RJ0 1/20 0.61
OPRK1 P41145 1/20 0.56
CYP2D6 P10635 1/20 0.56
ALOX15 P16050 1/20 0.56
GAA P10253 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538697 0.83 ALDH1A1 (0.74) ALDH1A1HTTKDM4EKMT2AMEN1
Hydrochloric Acid SCHEMBL9586835 0.82 ALDH1A1 (0.72) ALDH1A1HTTKDM4EKMT2AMEN1
SCHEMBL9537291 0.81 ALDH1A1 (0.71) ALDH1A1HTTKDM4EKMT2AMEN1
SCHEMBL9538032 0.81 MEN1 (0.69) ALDH1A1HTTKDM4EKMT2AMEN1
Hydrochloric Acid SCHEMBL9587817 0.81 ALDH1A1 (0.70) ALDH1A1HTTKDM4EKMT2AMEN1
SCHEMBL9588898 0.80 ALDH1A1 (0.90) ALDH1A1HTTKDM4EKMT2AMEN1
SCHEMBL9539965 0.80 ALDH1A1 (0.72) ALDH1A1HTTKDM4EKMT2AMEN1
SCHEMBL14355265 0.79 KMT2A (0.69) ALDH1A1HTTKDM4EKMT2AMEN1
Hydrochloric Acid SCHEMBL9589964 0.79 ALDH1A1 (0.71) ALDH1A1HTTKDM4EKMT2AMEN1
SCHEMBL3692842 0.78 KMT2A (1.00) ALDH1A1HTTKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5254595-A Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them ELF SANOFI (FR) 1993-10-19 US disclosed
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed