SCHEMBL9540063

SCHEMBL9540063

C=CCN1C(=O)Nc2ccc(Cl)cc2C1(CC1CC1)C1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
AKR1B1 P15121 3/20 0.34
PDE7A Q13946 1/20 0.33
MDM2 Q00987 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
TP53 P04637 1/20 0.33
IDO1 P14902 2/20 0.33
MAPT P10636 2/20 0.32
MAPK1 P28482 2/20 0.32
NR1I2 O75469 1/20 0.32
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
ADRB1 P08588 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CNR1 P21554 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540110 0.84 ELOVL6 (0.37) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9539021 0.80 AKR1B1 (0.48) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9540064 0.77 CYP46A1 (0.38) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9538999 0.75 AKR1B1 (0.49) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9539061 0.74 MEN1 (0.39) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9541633 0.72 PTGDR2 (0.44) PTGDR2CMA1
SCHEMBL9540069 0.71 MEN1 (0.41) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9539959 0.71 AKR1B1 (0.42) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL9539784 0.70 MEN1 (0.40) CYP46A1MEN1KMT2AAKR1B1PDE7A
SCHEMBL2473132 0.70 AKR1B1 (0.40) CYP46A1MEN1KMT2AAKR1B1PDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed