SCHEMBL9540110

SCHEMBL9540110

C=CCOCC1(C2CC2)c2cc(Cl)ccc2NC(=O)N1CC=C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELOVL6 Q9H5J4 2/20 0.37
CYP46A1 Q9Y6A2 2/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 2/20 0.32
MAPK1 P28482 2/20 0.32
NR1I2 O75469 1/20 0.32
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
ADRB1 P08588 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CNR1 P21554 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
AGTR1 P30556 1/20 0.32
CCKBR P32239 1/20 0.32
PPARG P37231 1/20 0.32
OPRK1 P41145 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539959 0.86 AKR1B1 (0.42) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9540063 0.84 CYP46A1 (0.36) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9539091 0.78 MEN1 (0.39) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9540011 0.74 ELOVL6 (0.35) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9539784 0.74 MEN1 (0.40) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9540146 0.74 PTGDR2 (0.42) PTGDR2
SCHEMBL9538999 0.73 AKR1B1 (0.49) CYP46A1MEN1KMT2AMAPTMAPK1
SCHEMBL9541557 0.72 MEN1 (0.38) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9540069 0.71 MEN1 (0.41) ELOVL6CYP46A1MEN1KMT2AMAPT
SCHEMBL9539957 0.69 AKR1B1 (0.47) ELOVL6CYP46A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed