SCHEMBL9540073

SCHEMBL9540073

CC(C)N1C(=O)Nc2ccc(Cl)cc2C1(O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
IDO1 P14902 2/20 0.42
AKR1B1 P15121 3/20 0.40
MAPT P10636 1/20 0.39
PGR P06401 1/20 0.37
CHRM1 P11229 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541565 0.84 AKR1B1 (0.51) MEN1KMT2AIDO1AKR1B1MAPT
SCHEMBL9539014 0.81 AKR1B1 (0.40) MEN1KMT2AIDO1AKR1B1MAPT
SCHEMBL11388713 0.81 MDM2 (0.46) MEN1KMT2AIDO1AKR1B1
SCHEMBL11882562 0.80 MDM2 (0.54) MEN1KMT2AIDO1AKR1B1
SCHEMBL9542678 0.79 AKR1B1 (0.38) MEN1KMT2AIDO1AKR1B1MAPT
SCHEMBL27311876 0.78 MDM2 (0.55) MEN1KMT2AIDO1MAPT
SCHEMBL9539948 0.77 KDM4E (0.52) MEN1KMT2AIDO1AKR1B1MAPT
SCHEMBL9540193 0.75 MEN1 (0.47) MEN1KMT2AIDO1AKR1B1MAPT
SCHEMBL2474367 0.75 MDM2 (0.41) MEN1KMT2AIDO1MAPT
SCHEMBL9539002 0.73 SCN9A (0.47) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed