SCHEMBL9539002

SCHEMBL9539002

COc1ccc(CN2C(=O)Nc3ccc(Cl)cc3C2(O)c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.47
MDM2 Q00987 9/20 0.46
CBX7 O95931 1/20 0.44
CDYL Q9Y232 1/20 0.44
ADAMTS5 Q9UNA0 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
CCR2 P41597 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRL1 P41146 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27311876 0.89 MDM2 (0.55) SCN9AMDM2TP53MAPT
SCHEMBL11882562 0.83 MDM2 (0.54) MDM2CBX7CDYL
SCHEMBL9539179 0.82 ADAMTS5 (0.42) SCN9AMDM2CBX7CDYLADAMTS5
SCHEMBL11388713 0.82 MDM2 (0.46) MDM2CBX7CDYL
SCHEMBL9540109 0.82 TP53 (0.43) SCN9AMDM2CBX7CDYLADAMTS5
SCHEMBL30877037 0.77 HSD11B1 (0.48) MDM2PTGDR2
SCHEMBL27311873 0.77 HSD11B1 (0.48) MDM2PTGDR2
SCHEMBL2474367 0.77 MDM2 (0.41) MDM2MAPT
SCHEMBL9541565 0.75 AKR1B1 (0.51) MDM2MAPT
SCHEMBL1819302 0.75 MDM2 (0.82) SCN9AMDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed