SCHEMBL9540087

SCHEMBL9540087

COc1ccc([N+](=O)[O-])c(NCc2ccccn2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.58
KMT2A Q03164 5/20 0.50
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 1/20 0.50
PKM P14618 3/20 0.49
RAB9A P51151 2/20 0.49
AKR1B10 O60218 1/20 0.49
AKR1B1 P15121 1/20 0.49
AKR1C4 P17516 1/20 0.49
AKR1C3 P42330 1/20 0.49
AKR1C2 P52895 1/20 0.49
AKR1C1 Q04828 1/20 0.49
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
ALPG P10696 1/20 0.48
VNN1 O95497 1/20 0.48
LMNA P02545 1/20 0.48
MEN1 O00255 4/20 0.48
BCHE P06276 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538655 0.91 CTSB (0.58) CTSBKMT2AALDH1A1NPC1PKM
SCHEMBL14247323 0.81 CTSB (0.61) CTSBKMT2AALDH1A1NPC1PKM
SCHEMBL18547825 0.81 CTSB (0.61) CTSBKMT2AALDH1A1PKMMAPT
SCHEMBL6474847 0.81 HTR6 (0.58) KMT2AALDH1A1NPC1AKR1B10AKR1B1
SCHEMBL7322890 0.81 CTSB (0.66) CTSBKMT2AALDH1A1NPC1PKM
SCHEMBL17714697 0.80 KMT2A (0.53) KMT2AALDH1A1NPC1RAB9AMAPT
SCHEMBL16407609 0.79 NPC1 (0.53) KMT2AALDH1A1NPC1RAB9AAKR1B10
SCHEMBL11037162 0.79 KMT2A (0.52) KMT2AALDH1A1NPC1RAB9AMAPT
SCHEMBL4309629 0.78 MAPT (0.62) KMT2AALDH1A1NPC1RAB9AAKR1B10
SCHEMBL23144814 0.78 MAPT (0.60) KMT2AALDH1A1NPC1RAB9AAKR1B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3022196-B1 NOVEL BENZIMIDAZOLIUM COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-09-06 EP disclosed
US-9328131-B2 Benzimidazolium compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-05-03 US disclosed
WO-2015007519-A1 NOVEL BENZIMIDAZOLIUM COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-01-22 WO disclosed
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed