SCHEMBL9540133

SCHEMBL9540133

CN(C)CC1(c2ccccc2)c2cc(Cl)ccc2NC(=S)N1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 7/20 0.39
AKR1B1 P15121 3/20 0.36
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
SLC6A2 P23975 2/20 0.35
CHRM1 P11229 4/20 0.34
MEN1 O00255 2/20 0.34
TP53 P04637 2/20 0.34
CYP3A4 P08684 2/20 0.34
KMT2A Q03164 2/20 0.34
SLC22A1 O15245 1/20 0.34
ABCB11 O95342 1/20 0.34
CYP1A2 P05177 1/20 0.34
ADRB2 P07550 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
ADRB1 P08588 1/20 0.34
HTR1A P08908 1/20 0.34
CHRM5 P08912 1/20 0.34
ADRA2A P08913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540047 0.88 PGR (0.40) PGRAKR1B1CHRM1MEN1KMT2A
SCHEMBL9539805 0.86 PGR (0.41) PGRAKR1B1CHRM1MEN1KMT2A
SCHEMBL9539937 0.84 CHRM1 (0.41) PGRAKR1B1CHRM1MEN1KMT2A
SCHEMBL9539997 0.83 PGR (0.39) PGRAKR1B1CHRM1CYP2D6MAPT
SCHEMBL9539803 0.82 PGR (0.38) PGRAKR1B1CHRM1OPRM1KDM4E
SCHEMBL9540169 0.82 IDO1 (0.41) PGRAKR1B1MEN1TP53KMT2A
SCHEMBL9540123 0.82 PGR (0.43) PGRAKR1B1CHRM1MEN1KMT2A
SCHEMBL9541572 0.80 PGR (0.37) PGRAKR1B1CHRM1MEN1KMT2A
SCHEMBL9539988 0.79 PGR (0.36) PGRAKR1B1CHRM1OPRM1MAPT
SCHEMBL9542738 0.79 PGR (0.36) PGRAKR1B1CHRM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed