SCHEMBL9540169

SCHEMBL9540169

CN1C(=S)Nc2ccc(Cl)cc2C1(CC(=O)O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.41
PGR P06401 3/20 0.38
AKR1B1 P15121 4/20 0.38
CBX7 O95931 2/20 0.36
CDYL Q9Y232 2/20 0.36
CDYL2 Q8N8U2 1/20 0.36
CDY1; CDY1B Q9Y6F8 1/20 0.36
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
HSD11B1 P28845 1/20 0.34
EPHX2 P34913 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540148 0.86 IDO1 (0.37) IDO1PGRAKR1B1CBX7CDYL
SCHEMBL9539805 0.85 PGR (0.41) PGRAKR1B1MEN1KMT2A
SCHEMBL9539997 0.84 PGR (0.39) IDO1PGRAKR1B1EPHX2
SCHEMBL9540047 0.84 PGR (0.40) IDO1PGRAKR1B1MEN1KMT2A
SCHEMBL9539937 0.83 CHRM1 (0.41) PGRAKR1B1MEN1KMT2A
SCHEMBL9540133 0.82 PGR (0.39) PGRAKR1B1TP53MEN1KMT2A
SCHEMBL9541572 0.81 PGR (0.37) IDO1PGRAKR1B1MEN1KMT2A
SCHEMBL9539803 0.81 PGR (0.38) PGRAKR1B1
SCHEMBL9540123 0.81 PGR (0.43) IDO1PGRAKR1B1MEN1KMT2A
SCHEMBL9539988 0.81 PGR (0.36) IDO1PGRAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed