SCHEMBL9540922

SCHEMBL9540922

CCOC(=O)c1c(SC)nc2sc3ccccc3n2c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.53
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
ALDH1A1 P00352 5/20 0.46
MAPT P10636 5/20 0.46
HPGD P15428 5/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
RAB9A P51151 1/20 0.45
HSD17B10 Q99714 1/20 0.45
L3MBTL1 Q9Y468 5/20 0.43
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
POLB P06746 3/20 0.43
CTDSP1 Q9GZU7 2/20 0.43
TDP1 Q9NUW8 2/20 0.41
HCRTR1 O43613 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543555 0.85 CYP1A2 (0.65) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL9539886 0.83 KDM4E (0.54) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL10463716 0.75 KDM4E (0.51) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL9542451 0.72 MAPK1 (0.56) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL3445304 0.71 MAPT (0.42) KDM4EALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL7331553 0.70 KDM4E (0.51) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL10464594 0.69 KDM4E (0.47) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL13317085 0.69 KDM4E (0.60) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL10931099 0.68 EGFR (0.51) KDM4ECYP1A2CYP2C9ALDH1A1MAPT
SCHEMBL2922603 0.68 GAA (0.53) KDM4ECYP1A2ALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013664-A2 BIHETEROCYCLIC FUNGICIDAL COMPOUNDS SCHERING AGROCHEMICALS LIMITED (GB) 1993-07-22 WO disclosed