SCHEMBL9540987

SCHEMBL9540987

C=CCN(C=O)c1ccc(Br)cc1CCC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.35
GPR17 Q13304 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
SLC6A2 P23975 1/20 0.33
ADRA1D P25100 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR1E P28566 1/20 0.33
SLC6A4 P31645 1/20 0.33
HTR7 P34969 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541015 0.72 AKR1B1 (0.43) NPSR1ADRA1AMAPTALDH1A1HPGD
SCHEMBL9541026 0.69 LTB4R (0.40) PDPK1PTGDR2FFAR4
SCHEMBL19865372 0.69 HPGD (0.50) GPR17NPSR1PTGDR2FFAR1FFAR4
SCHEMBL7544691 0.68 PTGDR2 (0.41) HTR1AADRA2ADRD2ADRA2BADRA2C
SCHEMBL28387747 0.67 PTGDR2 (0.53) PDPK1GPR17NPSR1PTGDR2FFAR1
SCHEMBL14430303 0.67 PDPK1 (0.47) PDPK1GPR17NPSR1PTGDR2FFAR1
SCHEMBL18397695 0.67 APEX1 (0.51) GPR17NPSR1PTGDR2KEAP1FFAR1
SCHEMBL29604377 0.67 PDPK1 (0.47) PDPK1GPR17NPSR1PTGDR2FFAR1
SCHEMBL31690287 0.67 NPSR1 (0.44) GPR17NPSR1PTGDR2FFAR1FFAR4
SCHEMBL28651618 0.66 NPSR1 (0.47) PDPK1GPR17NPSR1PTGDR2KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed