SCHEMBL9541015

SCHEMBL9541015

C=CCN(C=O)c1ccccc1CC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.43
TDP1 Q9NUW8 1/20 0.39
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
BCAT2 O15382 1/20 0.36
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CXCL8 P10145 5/20 0.35
CYP1A2 P05177 1/20 0.34
PTGS2 P35354 2/20 0.34
AKR1B10 O60218 1/20 0.33
UGT1A9 O60656 1/20 0.33
TRPA1 O75762 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10434660 0.76 C5AR1 (0.36) KDM4EMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL11406694 0.73 CXCL8 (0.44) AKR1B1TDP1CYP2C9SMN1; SMN2CXCL8
SCHEMBL9540987 0.72 PDPK1 (0.35) HPGDKDM4EMAPTALDH1A1NPSR1
SCHEMBL11415456 0.72 CXCL8 (0.45) AKR1B1TDP1CYP2C9SMN1; SMN2CXCL8
SCHEMBL11412753 0.72 CXCL8 (0.43) AKR1B1TDP1CYP2C9SMN1; SMN2CXCL8
SCHEMBL11418236 0.72 CXCL8 (0.43) AKR1B1TDP1CYP2C9SMN1; SMN2CXCL8
SCHEMBL9064675 0.72 C5AR1 (0.36) KDM4EMEN1KMT2ASMN1; SMN2POLB
SCHEMBL28211714 0.72 AKR1B1 (0.46) AKR1B1TDP1BCAT2KDM4EMAPT
SCHEMBL277886 0.71 ESR1 (0.42) HPGDKDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL29959951 0.71 ESR1 (0.42) HPGDKDM4EMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed