SCHEMBL9541241

SCHEMBL9541241

Cc1cccc2c1N(CC(N)=O)C(=O)C(N)CC2c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 7/20 0.47
CYP2C19 P33261 2/20 0.42
SIGMAR1 Q99720 2/20 0.38
AADAT Q8N5Z0 1/20 0.38
RAB9A P51151 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KMT2A Q03164 2/20 0.34
KIF11 P52732 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
AMPD2 Q01433 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922827 0.89 CCKBR (0.47) CCKBRCYP2C19SIGMAR1RAB9ASLC6A2
SCHEMBL8919181 0.86 CCKBR (0.63) CCKBR
SCHEMBL8920848 0.82 CYP2C19 (0.47) CCKBRCYP2C19SIGMAR1RAB9AKMT2A
SCHEMBL8398546 0.81 CCKBR (0.48) CCKBR
SCHEMBL9544058 0.79 CCKBR (0.47) CCKBRCYP2C19SIGMAR1AADATKMT2A
SCHEMBL9541664 0.79 CCKBR (0.48) CCKBRCYP2C19
SCHEMBL9541509 0.78 CCKBR (0.68) CCKBR
SCHEMBL8402157 0.78 CCKBR (0.50) CCKBRCYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL9543807 0.76 CCKBR (0.80) CCKBR
SCHEMBL8398551 0.76 CYP2C19 (0.41) CCKBRCYP2C19AADATTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed